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Counerotte Stéphane

Département de pharmacie

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Main Referenced Co-authors
Pirotte, Bernard  (22)
Foidart, Jean-Michel  (13)
Kempen, I. (12)
De Tullio, Pascal  (11)
Noël, Agnès  (10)
Main Referenced Keywords
Anti-cancer (1); Antimalarial Medicines (1); Cancer (1); Cell invasion (1); cell invasion (1);
Main Referenced Unit & Research Centers
Centre Interfacultaire de Recherche du Médicament - CIRM (2)
Main Referenced Disciplines
Pharmacy, pharmacology & toxicology (22)
Oncology (1)
Biochemistry, biophysics & molecular biology (1)

Publications (total 24)

The most downloaded
618 downloads
Kempen, I., Hemmer, M., Counerotte, S., Pochet, L., De Tullio, P., Foidart, J.-M., Blacher, S., Noël, A., Frankenne, F., & Pirotte, B. (December 2008). 6-Substituted 2-Oxo-2h-1-Benzopyran-3-Carboxylic Acid Derivatives in a New Approach of the Treatment of Cancer Cell Invasion and Metastasis. European Journal of Medicinal Chemistry, 43 (12), 2735-50. doi:10.1016/j.ejmech.2008.01.024 https://hdl.handle.net/2268/9663

The most cited

103 citations (Scopus®)

Kempen, I., Papapostolou, D., Thierry, N., Pochet, L., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Noël, A., & Pirotte, B. (07 April 2003). 3-Bromophenyl 6-acetoxymethyl-2-oxo-2H-1-benzopyran-3-carboxylate inhibits cancer cell invasion in vitro and tumour growth in vivo. British Journal of Cancer, 88 (7), 1111-1118. doi:10.1038/sj.bjc.6600856 https://hdl.handle.net/2268/12351

Habyalimana, V., Mbinze Kindenge, J., Kalenda Tshilombo, N., Dispas, A., Yemoa Loconon, A., Sacre, P.-Y., Widart, J., De Tullio, P., Counerotte, S., Kadima Ntokamunda, J.-L., Ziemons, E., Hubert, P., & Marini Djang'Eing'A, R. (02 December 2015). Analytical Tools and Strategic Approach to Detect Poor Quality Medicines, Identify Unknown Components, and Timely Alerts for Appropriate Measures: Case Study of Antimalarial Medicines. American Journal of Analytical Chemistry, 6, 977-994. doi:10.4236/ajac.2015.613093
Peer reviewed

Habyalimana, V., Dispas, A., Sacre, P.-Y., Widart, J., De Tullio, P., Counerotte, S., Kadima, N. J., Ziemons, E., Hubert, P., & Marini Djang'Eing'A, R. (28 May 2015). USE OF SIMPLE AND COMPLEX ANALYTICAL TOOLS TO DETECT POOR QUALITY MEDICINES: CASE OF RWANDA [Paper presentation]. 18th Forum of Pharmaceutical Sciences, Blankenberge, Belgium.

DUBOIS, N., Counerotte, S., Goffin, E., Pirotte, B., & Charlier, C. (April 2014). Validation analytique d'une méthode chromatographique destinée à rechercher et à identifier les opiacés naturels ou (semi) synthétiques. Annales de Biologie Clinique, 72 (2), 197-206. doi:10.1684/abc.2014.0944
Peer Reviewed verified by ORBi

Kempen, I., Hemmer, M., Counerotte, S., Pochet, L., De Tullio, P., Foidart, J.-M., Blacher, S., Noël, A., Frankenne, F., & Pirotte, B. (December 2008). 6-Substituted 2-Oxo-2h-1-Benzopyran-3-Carboxylic Acid Derivatives in a New Approach of the Treatment of Cancer Cell Invasion and Metastasis. European Journal of Medicinal Chemistry, 43 (12), 2735-50. doi:10.1016/j.ejmech.2008.01.024
Peer Reviewed verified by ORBi

Francotte, P., De Tullio, P., Fraikin, P., Counerotte, S., Goffin, E., Danober, L., Lestage, P., Renard, P., Caignard, D. H., & Pirotte, B. (17 May 2008). Design, synthesis and pharmacological evaluation of novel 7-substituted 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxides acting as AMPA potentiators [Poster presentation]. Réunion de la Société Belge de Physiologie et de Pharmacologie Fondamentales et Cliniques, Liège, Belgium.

Francotte, P., Fraikin, P., De Tullio, P., Graindorge, E., Dintilhac, G., Counerotte, S., Goffin, E., Danober, L., Lestage, P., Lesur, B., Caignard, D. H., & Pirotte, B. (May 2007). Design, synthèse et évaluation pharmacologique de 1,2,4-thiénothiadiazine 1,1-dioxydes en tant que nouveaux potentialisateurs AMPA [Poster presentation]. 21èmes Journées Franco-Belges de Pharmacochimie, Namur, Belgium.

Francotte, P., De Tullio, P., Fraikin, P., Counerotte, S., Goffin, E., Danober, L., Lestage, P., Renard, P., Caignard, D. H., & Pirotte, B. (August 2006). Design, synthesis and pharmacological evaluation of novel 7-substituted 3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxides acting as AMPA potentiators [Poster presentation]. XIXth International Symposium on Medicinal Chemistry, Istanbul, Turkey.

Francotte, P., Fraikin, P., De Tullio, P., Counerotte, S., Goffin, E., Danober, L., Lestage, P., Renard, P., Caignard, D. H., & Pirotte, B. (June 2006). Design, synthèse et évaluation pharmacologique de 1,2,4-pytridothiadiazine 1,1-dioxydes en tant que nouveaux potentiateurs AMPA [Poster presentation]. 20èmes Journées Franco-Belges de Pharmacochimie, Lille, France.

Pirotte, B., Counerotte, S., Detry, V., Frankenne, F., Foidart, J.-M., & Noël, A. (02 March 2006). Preparation of 5-(1,1'-biphenyl)-4-yl-5-(4-(4-aminoacylphenyl)-piperazin)-1-yl-pyrimidine-2,4,6-triones and their use as inhibitors of zinc metalloendopeptidases.

De Tullio, P., Dupont, L., Francotte, P., Counerotte, S., Lebrun, P., & Pirotte, B. (2006). Three-Dimentional Quantitative Structure-Activity Relationships of ATP-Sensitive Potassium (KATP) Channel Openers Belonging to the 3-Alkylamino-4H-1,2,4-benzo- and 3-Alkylamino-4H-1,2,4-pyridothiadiazine 1,1-Dioxide Families. Journal of Medicinal Chemistry, 49, 6779-6788. doi:10.1021/jm060534w
Peer Reviewed verified by ORBi

Francotte, P., De Tullio, P., Fraikin, P., Counerotte, S., Goffin, E., & Pirotte, B. (2006). In Search of Novel Ampa Potentiators. Recent Patents on CNS Drug Discovery, 1 (3), 239-46. doi:10.2174/157488906778773661
Peer reviewed

Boverie, S., Antoine, M.-H., Somers, F., Becker, B., Sebille, S., Ouedraogo, R., Counerotte, S., Pirotte, B., Lebrun, P., & De Tullio, P. (2005). Effect on KATP channel activation properties and tissue selctivity of the nature of the substituent in the 7- and the 3-position of 4H-1,2,4-benzothiadiazine. Journal of Medicinal Chemistry, 48, 3492-3503. doi:10.1021/jm0311339
Peer Reviewed verified by ORBi

De Tullio, P., Boverie, S., Becker, B., Antoine, M.-H., Nguyen, Q.-A., Francotte, P., Counerotte, S., Sebille, S., Pirotte, B., & Lebrun, P. (2005). 3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxides as ATP-sensitive potassium channel openers : effect of 6,7-distribution on potency and tissue selectivity. Journal of Medicinal Chemistry, 48, 4990-5000. doi:10.1021/jm0580050
Peer Reviewed verified by ORBi

Kempen, I., Counerotte, S., Frankenne, F., Noël, A., Foidart, J.-M., & Pirotte, B. (2004). Effects of recently developed 6-substituted 3-bromophenyl 2-oxo-2H-1-benzopyran-3-carboxylate derivatives on HT1080 cell invasion in vitro. Fundamental and Clinical Pharmacology, 271.
Peer Reviewed verified by ORBi

Kempen, I., Counerotte, S., Frankenne, F., Noël, A., Foidart, J.-M., & Pirotte, B. (22 November 2003). Effects of recently developed 6-substituted 3-bromophenyl 2-oxo-2H-1-benzopyran-3-carboxylate derivatives on HT1080 cell invasion in vitro [Poster presentation]. Réunion de la Société Belge de Physiologie et de Pharmacologie Fondamentales et Cliniques, Liège, Belgium.

Kempen, I., Counerotte, S., Frankenne, F., Foidart, J.-M., Noël, A., & Pirotte, B. (May 2003). Anti-invasive and anti-migrative properties of recently developed 6-substituted 2-oxo-2H-1-benzopyran-3-carboxylic acid derivatives [Poster presentation]. 11th Forum of pharmaceutical sciences, Spa, Belgium.

Kempen, I., Papapostolou, D., Thierry, N., Pochet, L., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Noël, A., & Pirotte, B. (07 April 2003). 3-Bromophenyl 6-acetoxymethyl-2-oxo-2H-1-benzopyran-3-carboxylate inhibits cancer cell invasion in vitro and tumour growth in vivo. British Journal of Cancer, 88 (7), 1111-1118. doi:10.1038/sj.bjc.6600856
Peer Reviewed verified by ORBi

Kempen, I., Counerotte, S., Frankenne, F., Foidart, J.-M., Noël, A., & Pirotte, B. (31 January 2003). Les esters du 6-hydroxymethyl-2-oxo-2H-1-benzopyrane-3-carboxylate de 3-bromophényle inhibent l’invasion des cellules de fibrosarcome humain in vitro [Poster presentation]. 10ème Journée Jeunes Chercheurs, Paris, France.

Kempen, I., Counerotte, S., Frankenne, F., Noël, A., Foidart, J.-M., & Pirotte, B. (May 2002). Les esters du 6-hydroxyméthyl-2-oxo-2H-1-benzopyrane-3-carboxylate de 3-bromophényle en tant qu’agents inhibiteurs de l’invasion cellulaire in vitro [Poster presentation]. XVIemes Journées Franco-Belges de Pharmacochimie, Bagnoles de l’Orne, France.

Kempen, I., Counerotte, S., Frankenne, F., Foidart, J.-M., & Pirotte, B. (25 January 2002). Synthèse et évaluation pharmacologique de dérivés de l'acide 2-oxo-2H-1-benzopyrane-3-carboxylique en tant qu'agents inhibiteurs de l'invasion cellulaire in vitro [Poster presentation]. Journée Jeunes Chercheurs, Paris, France.

Kempen, I., Pochet, L., Papapostolou, D., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Frankenne, F., & Pirotte, B. (16 October 2001). Effects on in vitro and in vivo cellular invasion of two 6-(acetoxymethyl)-2-oxo-2H-1-benzopyran-3-carboxylic acid derivatives [Poster presentation]. Molecular Mechanisms in Cancer and Alzheimer’s disease, Bruxelles, Belgium.

Kempen, I., Pochet, L., Papapostolou, D., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Frankenne, F., & Pirotte, B. (01 June 2001). Comparaison de l’effet de deux dérivés de l’acide 6-(acetoxymethyl)-2-oxo-2H-1-benzopyrane-3-carboxylique sur l’inhibition de l’invasion cellulaire in vitro et in vivo [Poster presentation]. XVémes Journées Franco-Belges de Pharmacochimie, Namur, Belgium.

Kempen, I., Papapostolou, D., Pochet, L., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Noël, A., & Pirotte, B. (May 2001). Effects on cellular invasion of two synthetic coumarins [Paper presentation]. 10th Forum of Pharmaceutical Sciences, Montréal, Canada.

Kempen, I., Pochet, L., Papapostolu, D., Counerotte, S., Masereel, B., Foidart, J.-M., Reboud-Ravaux, M., Noël, A., & Pirotte, B. (21 April 2001). Effects on cellular invasion of 6-(acetoxymethyl)-2-oxo-2H-1-benzopyran-3-carboxylic acid derivatives [Poster presentation]. Spring Meeting Angiogenesis, Liège, Belgium.

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